11.1 Prescribing and administering

11.2 Control of microbial contamination

11.3.1 Antibacterials

11.3.2 Antifungals

11.3.3 Antivirals

11.4.1 Corticosteroids

11.4.2 Other anti‑inflammatory preparations

11.5 Mydriatics and cycloplegics

11.6 Glaucoma

11.7 Local anaesthetics

11.8.1 Tear deficiency

11.8.2.1 Ocular diagnostic preparations
11.8.2.2 Subfoveal choroidal neovascularisation

11.8.2.3 Chemical burns

11.8.2.4 Other preparations

11.9 Contact lenses

 

11.1 Prescribing and administering

A prescription for eye preparations should specify if a separate bottle is needed for each eye and if preservative free drops or single dose units are required.  It should be specified whether the right, left or both eyes are to be treated. The abbreviations RE, LE and R+L may be used but not BE because of potential confusion. For outpatient prescriptions a stop date is needed if treatment is to finish before the next visit.
For all eye drops the recommended dose is one drop because of the limited size of the conjunctival sac. If different drops are to be given at the same time of day there should be an interval of about 3 mins between treatments. Preparations that sting should be given last. Systemic absorption via the nasal mucosa may be a problem with some drugs, eg beta blockers or adrenaline, and this can be minimised by compressing the lacrimal sac at the medial canthus for 1min during and after administration.
Preservative-free eye drops should be considered: (i) when a patient becomes ‘sensitive’ to preservatives, (ii) in order to lessen the preservative load when a patient is using a considerable number of eye drops (ie more than three), (iii) in the short term where inflammation (eg allergic conjunctivitis) makes it difficult to detect an adverse effect of the preservative in the additional eye drops.
Various aids can help the elderly or handicapped to give their own eye drops and details are available at the Pharmacy.
Eye ointments are used for local treatment of lids, for prolonged treatment at night and to reduce the number of drops given. If drops and ointment are used at the same time, drops should be given first.

11.2 Control of microbial contamination

All eye preparations are sterile when issued. They should be used with care to prevent contamination of contents and to avoid the spread of infection from one eye to the other.
For outpatients using multidose eye drops without preservative, 1 bottle is issued per week to treat one or both eyes. The bottle should be refrigerated and then discarded 7 days after opening. For multidose eye drops with preservative, 1 bottle per month is supplied to treat one or both eyes and this should be discarded 1 month after opening.
For inpatients fresh eye drops should be used on admission and after ophthalmic surgery. Each bottle should be labelled with the patient's forename and surname, the date opened and the eye(s) to be treated. One bottle should be used to treat both eyes except for antibiotic drops or when a separate bottle is specifically requested for each eye.
Preserved eye drops should be discarded after 14 days. Unpreserved drops should be stored in a refrigerator and discarded after 7 days.
All drops used in the operating theatres should be single use and if taken from a multidose container it should be discarded after single use. In the A&E department and outpatient clinics single use drops should be used whenever possible. Preserved drops in multidose containers may be reused but must be discarded after 12hrs in the A&E Dept and after each half day session in Outpatients. Drops should always be discarded after use in cases of suspected infection or if there is doubt about their quality.

11.3.1 Antibacterials

Ocular infections including conjunctivitis and blepharitis are best treated with chloramphenicol. If they fail to resolve quickly they should be referred to the Ophthalmology Dept. Combined antibiotic and steroid preparations are not recommended for non-specialist use.
First choices: Chloramphenicol eye drops: 0.5% [10ml £2.05].
Chloramphenicol eye ointment: 1.0% [4g £2.08].
Dose: For conjuctivitis the dose should vary according to severity. For severe infections 1 drop should be given every hour, reducing to 1 drop 4 times daily. Ointment should be considered for use at night. Treatment should be given until 48hrs after symptoms have resolved. For blepharitis the lid margins should be cleaned with cotton wool soaked in water and the ointment then massaged into the area 2-4 times daily.
Caution: Sensitivity to chloramphenicol, transient stinging with drops; aplastic anaemia occurs rarely.
For expert use:
Cefuroxime preservative-free eye drops:
5% [5ml £16.80].
Chloramphenicol single use eye drops: 0.5% [20 x 0.5ml £9.55].
Fusidic acid eye drops: 1% [5g £1.96].
Gentamicin eye drops: 0.3% (for Pseudomonas) [10ml £2.13].
Gentamicin Forte eye drops: 1.5% (Moorfields) [5ml £17.92].
Gentamicin Forte preservative-free eye drops: 1.5% (Moorfields) [5ml £18.73].
Ofloxacin eye drops: 0.3% [5ml, £2.17].
Penicillin preservative-free eye drops: 5,000 units/ml (for Strep, ophthalmia neonatorum). Prepared by NDDH pharmacy - unlicensed.
Propamidine eye drops: 0.1% (for acanthamoeba) [10ml £2.80]

11.3.2 Antifungals

Ocular mycosis requires expert treatment. Specialist eye drops from Moorfields are available at the Pharmacy.

11.3.3 Antivirals

First choice: Aciclovir eye ointment: 3% [4.5g £9.34]. Dose: for herpes simplex keratitis apply 5 times daily (every 4hrs) and continue for at least 3 days after healing is complete. Caution: Hypersensitivity to aciclovir; mild stinging after application; local irritation and inflammation. Steroid preparations should not be used in combination with antivirals.

11.4.1 Corticosteroids

Steroid eye drops are used for noninfected inflammatory conditions of the eye. They should usually be prescribed only after consultation with an ophthalmologist to minimise risk of masking an underlying condition, exacerbating an infection or causing steroid glaucoma. Dose frequency should vary according to the severity of inflammation, being tailed off gradually to avoid rebound inflammation.
Prednisolone 1% and dexamethasone 0.1% are about equivalent in potency.
Prednisolone, betamethasone and dexamethasone are readily absorbed and effective in treating internal inflammation; fluorometholone is absorbed to a lesser degree and has a mainly surface action.
First choice: Prednisolone eye drops: 0.5% [10ml £2.00]. Dose: 1 drop every 1-2hrs until control is achieved, then reduced gradually.
Caution: Systemic side effects may occur after prolonged use.
Other strengths of prednisolone:
Prednisolone eye drops: 1% (Pred-Forte®) [10ml £3.05].
Prednisolone eye drops: 0.1% (Moorfields) [10ml £10.84].
Prednisolone preservative free eye drops: 0.5% (Torbay) [10ml £3.65].
Prednisolone preservative free eye drops: 1% (Torbay) [10ml £3.70].
Prednisolone single use eye drops: 0.5% [20 x 0.5ml £10.08].
Other steroid preparations:
Betamethasone eye drops:
0.1% [10ml £2.23]. Dose and caution as for prednisolone.
Betamethasone eye ointment: 0.1% [3g £1.41].
For expert use:
Dexamethasone eye drops:
0.1% (Maxidex®) [5ml £1.42].
Dexamethasone preservative free eye drops: 0.1% (Moorfields) [8ml £7.90].
Dexamethasone single use eye drops: 0.1% [20 x 0.5ml £9.38].
Fluorometholone eye drops: 0.1% [5ml £1.71].

Corticosteroid eye preparations combined with antibiotics should be used only for post-operative inflammation when bacterial infection is likely.
For expert use:
Betamethasone 0.1% with neomycin 0.5% eye drops:
[10ml £2.32].
Maxitrol® eye drops: (dexamethasone + neomycin + polymyxin) [5ml £1.68].
Maxitrol® eye ointment: (dexamethasone + neomycin + polymyxin) [3.5g £1.44].
Prednisolone 0.5% with neomycin 0.5% eye drops: [10ml £2.00].
Caution: risk of neomycin toxicity at high doses.

Intravitreal corticosteroids

Link to NICE guidance

Dexamethasone intravitreal implant for the treatment of macular oedema secondary to retinal vein occlusion, TAG 229.

For expert use only:
Dexamethasone 700 microgram intravitreal implant: Ozurdex [£870.00].

11.4.2 Other anti-inflammatory preparations

First choice: Sodium cromoglicate eye drops: 2% [13.5ml £1.86].
Dose: for vernal catarrh and allergic conjuctivitis, 1 drop 4 times daily, or the ointment applied 2-3 times daily or at night. The full effect may develop over several days and treatment may be needed for the period of exposure to allergen. Caution: Allergy to preservative; transient nasal stinging.
Also:
Otrivine-Antistin® eye drops: [10ml £2.35].1 drop 2 or 3 times daily
For expert inpatient use:

11.5 Mydriatics and cycloplegics

First choice (for ocular examination): Tropicamide single use eye drops: 1% w/v [20 x 0.5ml £9.01]. Dose: 2 drops at 5min intervals with a further 1-2 drops after 30mins if needed (onset of action 20mins, duration 6-8hrs).
Caution: Photophobia may occur if the filtration angle is narrow; driving should be avoided until vision has returned to pre-treatment level.
For expert use:
Atropine sulphate eye drops:
1% [10ml £1.11].
Atropine sulphate single use eye drops: 1% [20 x 0.5ml £12.71].
Cyclopentolate eye drops: 0.5% [5ml £6.73] 1% [5ml £6.73].
Cyclopentolate single use eye drops: 0.5% & 1% [20 x 0.5ml £9.64].
Homatropine eye drops: 1% [10ml £2.57]; 2% [10ml £2.71].
Phenylephrine single use eye drops: 2.5% [20 x 0.5ml £9.53].
Phenylephrine eye drops: 10% [10ml £4.65].
Phenylephrine single use eye drops: 10% [20 x 0.5ml £9.53].
Tropicamide eye drops: 0.5% [5ml £1.29]; 1% [5ml £1.60].
Tropicamide single use eye drops: 0.5% & 1% [20 x 0.5ml £9.01].

11.6 Treatment of glaucoma

Link to NICE guidance

Diagnosis and management of glaucoma. Clinical Guideline No.85

 

Treatment for glaucoma should be started and changed by an ophthalmologist.

Beta blockers
First choice: Timolol eye drops
: 0.25% [5ml £1.53], 0.5%, [5ml £1.54].
Dose: initially 1 drop of 0.25% solution, increased to 0.5% if response is inadequate.
Also:
Timolol single use eye drops:
0.25% [30 x 0.2ml £8.45], 0.5% [30 x 0.2ml £9.65]
Betaxolol eye drops: 0.5% [5ml £1.90].

Caution: Ocular irritation, burning, itching and pain, decreased corneal sensitivity, diplopia and ptosis. Systemic absorption occurs and therefore beta-blocker eye drops are contra-indicated in patients with bradycardia, heart block or uncontrolled heart failure.
CSM Warning: The CSM has advised that beta-blockers, even those with apparent cardioselectivity, should not be used in patients with asthma or a history of obstructive airways disease, unless no alternative treatment is available. In such cases the risk of increasing bronchospasm should be appreciated and appropriate precautions taken.
For drug interactions see BNF Appendix 1.

Carbonic anhydrase inhibitors
Dorzolamide eye drops are used together with a topical beta-blocker, or alone if this is contra-indicated. Side effects are similar to those of systemic sulphonamides.
For expert use:
Dorzolamide
2%  eye drops: [5ml £5.88]. Dose: apply three times daily if used alone, twice daily if used with a topical beta-blocker.
Dorzolamide 2%  single use eye drops: [60 x 0.2ml £24.18]. Dose: apply three times daily if used alone, twice daily if used with a topical beta-blocker.
Dorzolamide 2% + timolol 0.5% eye drops: (Cosopt®) [5ml £9.06]. Dose: apply twice daily.
Dorzolamide 2% + timolol 0.5% eye drops single use eye drops: (Cosopt®) [60 x 0.2ml £28.59]. Dose: apply twice daily.
Also:
Brinzolamide eye drops:
1% (Azopt®) [5ml £6.56]. Dose: Apply twice a day, increasing to three times a day if necessary.
Also:
Acetazolamide tabs:
250mg [14 tabs £1.81]. Dose: 1-2 tabs initially then 1-4 tabs 4 times daily in divided doses.
Caution: Sensitivity to sulphonamides; renal failure and renal tubular acidosis; adrenal insufficiency; conditions with sodium or potassium depletion. Adverse effects include polydipsia, polyuria, potassium depletion, metabolic acidosis, crystalluria and renal calculi, paraesthesiae of extremities, anorexia and weight loss, rashes and rarely blood disorders.
Acetazolamide sustained release caps: 250mg [14 caps £7.77].
Acetazolamide injection: 500mg [£14.76].

Alpha2 adrenoreceptor agonists
Brimonidine, a selective alpha2-adrenoreceptor stimulant, is used for open-angle glaucoma and ocular hypertension when other drugs, particularly beta-blockers, are inappropriate.
For expert use:
Brimonidine eye drops:
0.2% [5ml £3.78]. Dose: one drop twice daily.

Prostaglandin analogues
Latanoprost are prostaglandin analogues which increase uveoscleral outflow. They are used to reduce intra-ocular pressure in ocular hypertension or in open-angle glaucoma if other drugs cannot control the condition adequately or are not tolerated. Patients should be monitored for any changes to eye coloration since an increase in the brown pigment in the iris may occur; particular care is required in those receiving treatment to one eye only.
First line:
Latanoprost eye drops:
0.005%: (Xalatan®) [2.5ml £12.48]. Dose: one drop daily.
Latanoprost eye drops: 0.005% + timolol 0.5%: (Xalacom®) [2.5ml £14.32]. Dose: one drop daily.
Second line:
For patients who cannot tolerate or who do reach target intraocular pressure with latanoprost.

Bimatoprost 0.03% eye drops: (Lumigan®) [3ml £10.30]. Dose: one drop daily.
For patients diagnosed as intolerant to eye preservatives
Tafluprost 0.0015% preservative free eye drops: (Saflutan®) [30 x 0.3ml £17.41]. Dose: one drop daily, preferably in the evening.

Miotics (cholinergics)
First choice: Pilocarpine eye drops: 0.5% [10ml £1.30]; 1% [10ml £2.82]; 2% [£2.77]; 3% [£1.55]; 4% [£3.60].
Pilocarpine single use eye drops: 2% [20 x 0.5ml £10.04].
Dose: 1 drop up to 4-6 times daily; for acute closed angle glaucoma pilocarpine 4% 1 drop every 5-15mins.
Caution: Ciliary spasm, cicatrizing conjuctivitis. Systemic absorption may cause sweating, bradycardia, intestinal colic, hypersalivation and bronchospasm.

11.7 Local anaesthetics

These are used for anaesthesia prior to tonometry, removal of foreign bodies, minor conjunctival and corneal surgery. Anaesthetised eyes should be padded to protect from dust and bacteria and patients should be advised not to touch their eyes for at least 30mins after a procedure. Anaesthetised eyes should be padded to protect them from dust and bacteria. If this is impracticable patients should be advised to avoid dust and not to touch their eyes for at least 30 minutes after a procedure.
First choice (for anaesthesia only): Proxymetacaine single use drops: 0.5% [20 x 0.5ml £9.51].
Also:
Oxybuprocaine single use drops:
0.4% [20 x 0.5ml £8.92].
Tetracaine single use eye drops: 0.5% & 1% (BAN = amethocaine) [20 x 0.5ml £8.93].
First choice (for anaesthesia with staining): Proxymetacaine 0.5% and fluorescein 0.25% single use drops: [20 x 0.5ml £10.59].

11.8.1 Tear deficiency

Artificial tears and lubricants are used for dry eye syndromes. Where troublesome mucus is present acetylcysteine may also help.
First choice: Hypromellose eye drops: 0.3% [10ml £1.60]. Dose: 1 drop as needed to relieve irritation or dryness. Caution: Prolonged and frequent use causes preservative toxicity in 9% of patients so those at risk should use preservative free drops. Different preparations vary in their osmolarity.
Also:
Acetylcysteine 5% without preservative eye drops:
(Moorfields) [10ml £14.41].
Carmellose single use drops: (Celluvisc®) 0.5% [30 x 0.4ml £5.75]; 1% [30 x 0.4ml £3.00].
Hypromellose preservative free eye drops: 0.3% (Moorfields) [30 x 0.4ml £4.60].
Polyvinyl alcohol eye drops: 1.4% (Sno Tears®) [10ml £1.06].
Simple eye ointment: [4g £3.22].
Lacri-lube® ointment: [3.5g £2.28].
Carbomer 0.2% liquid gel: (Viscotears®): [10g £2.94], preservative free [30 x 0.6ml £5.42].

11.8.2  Ocular diagnostic and perioperative preparations and photodynamic treatment

11.8.2.1 Ocular diagnostic preparations

First choice: Fluorescein sodium single use drops: 1% & 2%, [20 x 0.5ml £7.53]. Contact lenses, if worn, should be removed and 1 drop applied to damaged areas. Conjunctival abrasions stain yellow or orange, corneal abrasions or ulcers stain bright green and foreign bodies are surrounded by a green ring. Excess should be washed away with sodium chloride solution 0.9%.
Fluoret fluorescein strip: 1mg, for detecting corneal and conjunctival ulcers and epithelial defects. The strip is moistened with sterile sodium chloride solution 0.9% and the tip stroked across the conjunctiva with the eye looking down, after which the patient should blink several times [100 strips £5.92].
Vision Blue: [0.5ml syringe £16.50].

11.8.2.2 Subfoveal choroidal neovascularisation

Pegaptanib and ranibizumab are vascular endothelial growth factor inhibitors licensed for the treatment of neovascular (wet) age-related macular degeneration; they are given by intravitreal injection by specialists experienced in the management of this condition.

Link to NICE guidance

Macular degeneration (age related) ranibizimab & pegaptanib. No.155

For specialist use only
Ranibizumab solution for intravitreal injection: (Lucentis
®): 10mg/ml [0.23ml vial £761.20]. Dose: see BNF. NB antimicrobial eye drops should be administered into the affected eye for 3 days before and 3 days after each injection.

11.8.2.3 Chemical Burns

The cause of a chemical burn needs to be identified. The eye should be irrigated thoroughly until the fornices are neutral to universal indicator paper.
Sodium citrate eye drops: 10.11% (equivalent to citrate 6.5%), for acid and alkali burns (Moorfields) [10ml £17.55] Dose: 1 drop every 0.5-2hrs initially, the frequency reduced as needed but treatment continued until the epithelium has healed.
Potassium ascorbate eye drops: (equivalent to ascorbic acid 10%), eye drops are used in conjunction with sodium citrate drops at the same frequency (Moorfields) [10ml £16.82].


11.8.2.4 Other preparations

Operating theatre use:
Acetylcholine chloride injection:
(Miochol-E®) 1% [2ml £7.28].
Apraclonidine ophthalmic soln: (Iopidine®) 1% [0.25ml £3.24].
Balanced salt soln: [19ml £0.95; 500ml £2.50].
Flurbiprofen single use eye drops: 0.03% [40 x 0.4ml £37.15].
Hyaluronidase injection: 1500 units [£7.60].
Ketorolac eye drops: (Acular®) 0.5% [5ml £3.00].
Sodium hyaluronate injection: 10mg/ml [0.85ml £10.80].
Sodium hyaluronate injection: (GV) 14mg/ml [0.55ml £27.00].

Miscellaneous:
Apraclonidine eye drops: (Iopidine®) 0.5% [5ml £10.88].
Betamethasone sodium phosphate injection: 4mg in 1ml [£1.22].
Disodium edetate (EDTA) eye drops: 0.37% (Moorfields) [10ml £12.11].
Disodium edetate (EDTA) eye lotion: 0.37% (Moorfields) [20ml £55.67].
Sodium chloride eye drops:
0.9% [10ml £1.15]
Sodium chloride single use drops: 0.9% [20 x 0.5ml £6.80].
Sodium chloride eye drops: 5% (Torbay) [10ml £4.00].
Sodium chloride eye drops (unpreserved): 5% (Torbay) [10ml £4.78].
Zinc sulphate eye drops: 0.25% [10ml £3.78].
For expert use:
Botulinum toxin:
100 units (Botox®). [£138.20].
Botulinum toxin: 500 units (Dysport®). [£154.00].

11.9.1 Contact lenses

Contact lenses should be avoided during topical ocular therapy or should only be worn on medical advice. If they are worn, ointments and oily drops should not be used.
Soft lenses (hydrophilic) can absorb preservatives in eye drops causing irritation and sensitivity.
Drops containing benzalkonium chloride should never be used. Thiomersal is usually satisfactory and chlorhexidine rarely causes irritation.
Soft lenses may be stained by topical adrenaline, fluorescein, phenylephrine and Rose Bengal and by systemic phenolpthalein, rifampicin, sulphasalzine and tetracyclines.
Rigid lenses (hydrophobic) do not absorb preservatives but benzalkonium chloride can cause irritation. Rigid lenses with a hydrophilic surface should not come into contact with any solution containing benzalkonium chloride. Anti-inflammatory drops should not be used for prolonged periods.
Lubricants are available for hot dry eyes when contact lenses are used for medical reasons.
For papillary conjunctivitis induced by contact lenses:
Sodium cromoglicate eye drops 2% (see 11.4.2).

11.9.2 Primary care of contact lenses

Contact lens care products are only available from the hospital Ophthalmology Dept if lenses are fitted for medical reasons.
Soft lenses should be rinsed with sodium chloride solution 0.9% before wearing. Gas permeable and hard lenses should be wetted with 2 drops of polyvinyl alcohol 1.4% unless a wetting /soaking solution has been used.
For soft contact lenses:
Oxysept® 1 Step: [90 day pack £22.79].

For rigid gas permeable and hard contact lenses
Boston®  conditioning solution: [120ml £4.58].
Boston® cleaner: [30ml £4.58]
Total Care® disinfecting, storing and wetting solution: [120ml £4.57].
Total Care® daily cleaner: [30ml £4.42].

For all types of contact lenses
Amiclair® contact lens cleanser tabs: [24 tabs £5.58].
Lens Plus Ocupure® saline: [360ml £2.07].
Quattro® Multifunctional solution: [250ml £5.45]. NB 100ml starter pack available.